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A Nitrogen-Assisted One-Pot Heteroaryl Ketone Synthesis from Carboxylic Acids and Heteroaryl Halides

Krystyna Demkiw1, Hirofumi Araki2, Eric L Elliott1

  • 1Chemical Development Laboratories, Millennium Pharmaceuticals, Inc. , a subsidiary of Takeda Pharmaceutical Company Limited, 40 Landsdowne Street, Cambridge, Massachusetts 02139, United States.

The Journal of Organic Chemistry
|March 19, 2016
PubMed

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