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Updated: Sep 23, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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Simple and Expedient Access to Novel Fluorinated Thiazolo- and Oxazolo[3,2-a]pyrimidin-7-one Derivatives and Their

Wafa Blancou1,2, Badr Jismy1, Soufiane Touil2

  • 1Laboratoire de Physico-Chimie des Matériaux et des Electrolytes pour l'Energie (PCM2E), EA 6299, Avenue Monge, Faculté des Sciences, Université de Tours, Parc de Grandmont, 37200 Tours, France.

Molecules (Basel, Switzerland)
|May 14, 2022
PubMed

Keywords:
Sonogashira couplingSuzuki-Miyaurafluorinated alkynesone-pot reactionoxazolo[3,2-a]pyrimidin-7-onesregioselectivethiazolo[3,2-a]pyrimidin-7-ones

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