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Updated: Sep 2, 2025

Modification and Functionalization of the Guanidine Group by Tailor-made Precursors
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Development of subtype-selective covalent ligands for the adenosine A2B receptor by tuning the reactive group

Bert L H Beerkens1, Xuesong Wang1, Maria Avgeropoulou1

  • 1Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl.

RSC Medicinal Chemistry
|August 4, 2022
PubMed

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