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Updated: Jul 11, 2025

Constructing Cyclic Peptides Using an On-Tether Sulfonium Center
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Disulfide Click Reaction for Stapling of S-terminal Peptides

Qing Yu1, Leiyang Bai1, Xuefeng Jiang1,2,3

  • 1Shanghai Key Laboratory of Green Chemistry and Chemical Process, School of Chemistry and Molecular Engineering, East China Normal University, 3663 North Zhongshan Road, Shanghai, 200062, P. R. China.

Angewandte Chemie (International Ed. in English)
|November 11, 2023
PubMed

Keywords:
Cyclic PeptidesDisulfide Stapling ReagentsPeptide DeliveryReversible Staplingα-Helicity

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