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Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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N1-Selective Methylation of Pyrazoles via α-Halomethylsilanes as Masked Methylating Reagents

Emma Yang1, Derek M Dalton1

  • 1Department of Small Molecule Process Chemistry, Genentech, Inc., South San Francisco, California 94080, United States.

The Journal of Organic Chemistry
|February 29, 2024
PubMed

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