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Emerging approaches for antagonizing the aryl hydrocarbon receptor

Zdeněk Dvořák1, Sridhar Mani2, Jan Vondráček3

  • 1Department of Cell Biology and Genetics, Faculty of Science, Palacký University, Šlechtitelů 27, 783 71 Olomouc, Czech Republic.

Trends in Pharmacological Sciences
|June 6, 2025
PubMed
Summary

Developing novel aryl hydrocarbon receptor (AhR) antagonists is crucial. New strategies focus on selective targeting of AhR pathways and protein interactions for improved therapeutics.

Keywords:
AhR receptorallosteric modulationantagonismfunctional selectivity

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