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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Indole-based derivatives as anticancer agents: recent advances in structure-activity relationships and biological

Aashik Malik1, Mayank Yadav2, Jai Parkash Kadian3

  • 1Adarsh Vijendra Institute of Pharmaceutical Sciences, Shobhit University, Gangoh, 247001, Saharanpur, India. aashikmalik24@gmail.com.

Medicinal Chemistry Research : an International Journal for Rapid Communications on Design and Mechanisms of Action of Biologically Active Agents
|August 14, 2026
PubMed
Abstract

Keywords:
Anticancer agentsIndole derivativesMolecular hybridizationProtein kinasesStructure–activity relationshipTargeted therapy

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