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Bioorganic & Medicinal Chemistry Letters|December 1, 2015
Addressing cytotoxicity of 1,4-biphenyl amide derivatives: Discovery of new potent and selective 17β-hydroxysteroid dehydrogenase type 2 inhibitorsEmanuele Marco Gargano, Enrico Perspicace, Angelo Carotti, et al.Bioorganic & Medicinal Chemistry|July 1, 2008
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitorsFrancesco Leonetti, Marco Catto, Orazio Nicolotti, et al.Journal of Medicinal Chemistry|December 24, 2004
Design, synthesis, and 3D QSAR of novel potent and selective aromatase inhibitorsFrancesco Leonetti, Angelo Favia, Angela Rao, et al.European Journal of Medicinal Chemistry|September 27, 2014
Metabolic stability optimization and metabolite identification of 2,5-thiophene amide 17β-hydroxysteroid dehydrogenase type 2 inhibitorsEmanuele M Gargano, Enrico Perspicace, Nina Hanke, et al.ACS Chemical Neuroscience|September 24, 2014
First selective dual inhibitors of tau phosphorylation and Beta-amyloid aggregation, two major pathogenic mechanisms in Alzheimer's diseaseMarica Mariano, Christian Schmitt, Parisa Miralinaghi, et al.Farmaco (Societa Chimica Italiana : 1989)|February 13, 2003
Synthesis and biological evaluation of pyridazino[4,3-b]indoles and indeno[1,2-c]pyridazines as new ligands of central and peripheral benzodiazepine receptorsFrancesco Campagna, Fausta Palluotto, Maria Paola Mascia, et al.ALTEX|July 23, 2014
A k-NN algorithm for predicting the oral sub-chronic toxicity in the ratDomenico Gadaleta, Fabiola Pizzo, Anna Lombardo, et al.Journal of Computer-Aided Molecular Design|February 12, 2010
Screening of benzamidine-based thrombin inhibitors via a linear interaction energy in continuum electrostatics modelOrazio Nicolotti, Ilenia Giangreco, Teresa Fabiola Miscioscia, et al.Bioorganic & Medicinal Chemistry|March 12, 2003
Investigation of platelet aggregation inhibitory activity by phenyl amides and esters of piperidinecarboxylic acidsModesto de Candia, Luciana Summo, Antonio Carrieri, et al.Drug Discovery Today|July 8, 2014
REACH and in silico methods: an attractive opportunity for medicinal chemistsOrazio Nicolotti, Emilio Benfenati, Angelo Carotti, et al.Pageof 9