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Current Medicinal Chemistry
|
May 27, 2017
A Systematic Analysis of Physicochemical and ADME Properties of All Small Molecule Kinase Inhibitors Approved by US FDA from January 2001 to October 2015
Zhihong O Brien, Mehran F Moghaddam
Bioanalysis
|
January 12, 2017
Implementation of a novel ultra fast metabolic stability analysis method using exact mass TOF-MS
Joseph D Manna, Samantha J Richardson, Mehran F Moghaddam
Drug Metabolism Letters
|
February 24, 2016
Efficiency in Drug Discovery: Liver S9 Fraction Assay As a Screen for Metabolic Stability
Samantha J Richardson, April Bai, Ashutosh A Kulkarni, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals
|
December 18, 2001
Plasma pharmacokinetics and tissue distribution of a N-pyrrolo-[1,2-c]imidazolylphenyl sulfonamide in rats
Mehran F Moghaddam, Matthew S Bogdanffy, Alethia Brown, et al.
Drug Metabolism Letters
|
April 24, 2013
Application of 1D and 2D 1H-NMR in the structural elucidation of a N-glucuronidated metabolite and oxidized metabolites generated in microsomal incubation
Julius L Apuy, April Bai, David Paisner, et al.
Future Medicinal Chemistry
|
January 29, 2014
Proposing advancement criteria for efficient DMPK triage of new chemical entities
Ashutosh Kulkarni, Jennifer Riggs, Cindy Phan, et al.
Drug Metabolism Letters
|
April 10, 2009
Metabolite interference in pharmacokinetic studies
Mehran F Moghaddam, Jui-Hsiang Fan, Yang Tang, et al.
Drug Metabolism Letters
|
May 12, 2016
Formation of A Novel Purine Metabolite through CYP3A4 Bioactivation and Glutathione Conjugation
Julius L Apuy, Cathie Xiang, Sarah Franc, et al.
Drug Metabolism Letters
|
March 18, 2014
A proposed screening paradigm for discovery of covalent inhibitor drugs
Mehran F Moghaddam, Yang Tang, Zhihong O'Brien, et al.
Plos One
|
August 14, 2013
Pomalidomide shows significant therapeutic activity against CNS lymphoma with a major impact on the tumor microenvironment in murine models
Zhimin Li, Yushi Qiu, David Personett, et al.
Page
of 2
Search research articles
Search
Showing results (1-10 of 16) with videos related to
Sort By:
Page
of 2
Current Medicinal Chemistry
|
May 27, 2017
A Systematic Analysis of Physicochemical and ADME Properties of All Small Molecule Kinase Inhibitors Approved by US FDA from January 2001 to October 2015
Zhihong O Brien, Mehran F Moghaddam
Bioanalysis
|
January 12, 2017
Implementation of a novel ultra fast metabolic stability analysis method using exact mass TOF-MS
Joseph D Manna, Samantha J Richardson, Mehran F Moghaddam
Drug Metabolism Letters
|
February 24, 2016
Efficiency in Drug Discovery: Liver S9 Fraction Assay As a Screen for Metabolic Stability
Samantha J Richardson, April Bai, Ashutosh A Kulkarni, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals
|
December 18, 2001
Plasma pharmacokinetics and tissue distribution of a N-pyrrolo-[1,2-c]imidazolylphenyl sulfonamide in rats
Mehran F Moghaddam, Matthew S Bogdanffy, Alethia Brown, et al.
Drug Metabolism Letters
|
April 24, 2013
Application of 1D and 2D 1H-NMR in the structural elucidation of a N-glucuronidated metabolite and oxidized metabolites generated in microsomal incubation
Julius L Apuy, April Bai, David Paisner, et al.
Future Medicinal Chemistry
|
January 29, 2014
Proposing advancement criteria for efficient DMPK triage of new chemical entities
Ashutosh Kulkarni, Jennifer Riggs, Cindy Phan, et al.
Drug Metabolism Letters
|
April 10, 2009
Metabolite interference in pharmacokinetic studies
Mehran F Moghaddam, Jui-Hsiang Fan, Yang Tang, et al.
Drug Metabolism Letters
|
May 12, 2016
Formation of A Novel Purine Metabolite through CYP3A4 Bioactivation and Glutathione Conjugation
Julius L Apuy, Cathie Xiang, Sarah Franc, et al.
Drug Metabolism Letters
|
March 18, 2014
A proposed screening paradigm for discovery of covalent inhibitor drugs
Mehran F Moghaddam, Yang Tang, Zhihong O'Brien, et al.
Plos One
|
August 14, 2013
Pomalidomide shows significant therapeutic activity against CNS lymphoma with a major impact on the tumor microenvironment in murine models
Zhimin Li, Yushi Qiu, David Personett, et al.
Page
of 2