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Bioorganic & Medicinal Chemistry|March 13, 2019
The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitorsDavid N Deaton, Young Do, Jason Holt, et al.Bioorganic & Medicinal Chemistry|November 17, 2018
Design, synthesis and antifungal evaluation of borrelidin derivativesCaijuan Hu, Hao Su, Jinghan Luo, et al.Bioorganic & Medicinal Chemistry|November 19, 2018
Design, synthesis and in vitro evaluation of stilbene derivatives as novel LSD1 inhibitors for AML therapyYingchao Duan, Wenping Qin, Fengzhi Suo, et al.Bioorganic & Medicinal Chemistry|November 19, 2018
Dose dependent actions of LCL521 on acid ceramidase and key sphingolipid metabolitesAiping Bai, Alicja Bielawska, Mehrdad Rahmaniyan, et al.Bioorganic & Medicinal Chemistry|November 14, 2018
Syntheses of prodrug-type 2'-O-methyldithiomethyl oligonucleotides modified at natural four nucleoside residues and their conversions into natural 2'-hydroxy oligonucleotides under reducing conditionJunsuke Hayashi, Yosuke Ochi, Yasuyuki Morita, et al.Bioorganic & Medicinal Chemistry|November 14, 2018
Lobaric acid and pseudodepsidones inhibit NF-κB signaling pathway by activation of PPAR-γClaudia Carpentier, Xavier Barbeau, Jabrane Azelmat, et al.Bioorganic & Medicinal Chemistry|November 16, 2018
Modifying aroylhydrazone prochelators for hydrolytic stability and improved cytoprotection against oxidative stressQin Wang, Katherine J FranzBioorganic & Medicinal Chemistry|November 16, 2018
Screening, synthesis, crystal structure, and molecular basis of 6-amino-4-phenyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitriles as novel AKR1C3 inhibitorsXuehua Zheng, Zan Jiang, Xiaolin Li, et al.Bioorganic & Medicinal Chemistry|April 8, 2019
Proline-based hydroxamates targeting the zinc-dependent deacetylase LpxC: Synthesis, antibacterial properties, and docking studiesDmitrii V Kalinin, Oriana Agoglitta, Hélène Van de Vyver, et al.Bioorganic & Medicinal Chemistry|March 31, 2019
Effect of curcumin-nanoemulsion associated with photodynamic therapy in breast adenocarcinoma cell lineFrancielly Cristina Machado, Renata Prandini Adum de Matos, Fernando Lucas Primo, et al.Pageof 1,701