Emmanuel H Demont
14PUBLICATIONS
46CO-AUTHORS
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Publications (14)
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|Dec 30, 2025
BET Isoform Selectivity through Diverse Linkers for Bivalent Inhibitors: GSK785, a BRD2/4-Selective Bivalent BET Inhibitor.Francesco Rianjongdee, Stephen J Atkinson, Paul Bamborough
|Aug 20, 2021
Optimization of Naphthyridones into Selective TATA-Binding Protein Associated Factor 1 (TAF1) Bromodomain Inhibitors.Michael A Clegg, Natalie H Theodoulou, Paul Bamborough
|Aug 13, 2021
Discovery of a Novel Bromodomain and Extra Terminal Domain (BET) Protein Inhibitor, I-BET282E, Suitable for Clinical Progression.Katherine L Jones, Dominic M Beaumont, Sharon G Bernard
|Jul 14, 2021
Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors.Simon C C Lucas, Stephen J Atkinson, Chun-Wa Chung
|Jul 13, 2021
Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors.Jonathan T Seal, Stephen J Atkinson, Paul Bamborough
|Jul 12, 2021
Discovery of a Highly Selective BET BD2 Inhibitor from a DNA-Encoded Library Technology Screening Hit.Francesco Rianjongdee, Stephen J Atkinson, Chun-Wa Chung
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Frequent Collaborators
13 joint publications
Chun-Wa Chung
10 joint publications
Paul Bamborough
9 joint publications
Alex Preston
8 joint publications
Stephen J Atkinson
5 joint publications
Jonathan T Seal
3 joint publications
Lee A Harrison
3 joint publications
Francesco Rianjongdee
2 joint publications
Christopher Wellaway
2 joint publications
Nicholas C O Tomkinson
1 joint publications
Kallie Friston
