Malcolm P Huestis

7PUBLICATIONS
6CO-AUTHORS
Process control and simulationOrganic chemical synthesisF-block chemistryCheminformatics and quantitative structure-activity relationshipsOrganometallic chemistry
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Publications (7)

|Nov 09, 2022
Ni-Catalyzed Reductive Cross-Coupling of Cyclopropylamines and Other Strained Ring NHP Esters with (Hetero)Aryl Halides.

Michael S West, Alexis L Gabbey, Malcolm P Huestis

|Jan 28, 2022
Simple strategy towards amide bioisosteres.

Malcolm P Huestis, Jack A Terrett

|May 31, 2021
Targeting KRAS Mutant Cancers via Combination Treatment: Discovery of a Pyridopyridazinone pan-RAF Kinase Inhibitor.

Malcolm P Huestis, Matthew R Durk, Charles Eigenbrot

|Apr 28, 2021
Photoredox/Nickel Dual Catalytic Cross-Coupling of Potassium Thiomethyltrifluoroborates with Aryl and Heteroaryl Bromides.

Katherine Townsend, Malcolm P Huestis, John C Tellis

|Mar 29, 2021
Targeting KRAS Mutant Cancers via Combination Treatment: Discovery of a 5-Fluoro-4-(3H)-quinazolinone Aryl Urea pan-RAF Kinase Inhibitor.

Malcolm P Huestis, Darlene Dela Cruz, Antonio G DiPasquale

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