Niklas Papenkordt

7PUBLICATIONS
50CO-AUTHORS
Cheminformatics and quantitative structure-activity relationshipsBiologically active moleculesContaminant hydrologyMolecular targets
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Publications (7)

|May 05, 2026
Development of High-Affinity CHD1 Chromodomain Inhibitors.

|Oct 30, 2025
From Pharmacophore to Warhead: NAD+-Targeting Triazoles as Mechanism-Based Sirtuin Inhibitors.

Florian Friedrich, Marat Meleshin, Niklas Papenkordt

|Nov 11, 2024
Aromatic Amino Acid Hydroxylases as Off-Targets of Histone Deacetylase Inhibitors.

Anne Baumann, Niklas Papenkordt, Dina Robaa

|Oct 30, 2023
Development of First-in-Class Dual Sirt2/HDAC6 Inhibitors as Molecular Tools for Dual Inhibition of Tubulin Deacetylation.

Laura Sinatra, Anja Vogelmann, Florian Friedrich

|Jun 20, 2023
Melatonin-vorinostat hybrid ligands show higher histone deacetylase and cancer cell growth inhibition than vorinostat.

Youssef Y Helmi, Niklas Papenkordt, Georg Rennar

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