Facile reductive amination of aldehydes with electron-deficient anilines by acyloxyborohydrides in TFA: application

Eric E Boros1, James B Thompson, Subba R Katamreddy

  • 1GlaxoSmithKline Research & Development, Five Moore Drive, Research Triangle Park, North Carolina 27709, USA. eric.e.boros@gsk.com

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