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Updated: Jan 23, 2026

Identification of Mediators of T-cell Receptor Signaling via the Screening of Chemical Inhibitor Libraries
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Identification of a novel orally bioavailable ERK5 inhibitor with selectivity over p38α and BRD4

Stephanie M Myers1, Duncan C Miller1, Lauren Molyneux1

  • 1Newcastle Drug Discovery, Northern Institute for Cancer Research, School of Chemistry, Bedson Building, Newcastle University, Newcastle Upon Tyne, NE1 7RU, UK.

European Journal of Medicinal Chemistry
|June 19, 2019
PubMed

Keywords:
BMK1BioavailableERK5Extracellular regulated kinase 5KinasePyrrole carboxamide

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