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Updated: Aug 26, 2025

Facile Preparation of 4-Substituted Quinazoline Derivatives
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Dihydropyrazinoquinazolinones via SN2 Sulfamidate Ring-Opening and a Sequential Quinazolinone-Amidine Rearrangement

Jhewelle N Fitz-Henley1, Soren D Rozema1, Jennifer E Golden1

  • 1Division of Pharmaceutical Sciences, School of Pharmacy, University of Wisconsin─Madison, 777 Highland Avenue, Madison, Wisconsin 53705, United States.

The Journal of Organic Chemistry
|October 4, 2022
PubMed

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