Thomas G Davies

5PUBLICATIONS
21CO-AUTHORS
Molecular medicineBiologically active moleculesProteins and peptides
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Publications (5)

|Sep 10, 2026
The Discovery of GSK3227634: A Potent Inhaled Inhibitor of the KEAP1/NRF2 Protein-Protein Interaction for the Treatment of Chronic Obstructive Pulmonary Disease.

|Mar 11, 2024
Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase-2 (SHP2).

James E H Day, Valerio Berdini, Joan Castro

|Oct 27, 2021
Fragment-Guided Discovery of Pyrazole Carboxylic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2 Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction.

David Norton, William G Bonnette, James F Callahan

|Apr 12, 2019
Structure-Activity and Structure-Conformation Relationships of Aryl Propionic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1/Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1/NRF2) Protein-Protein Interaction.

Tom D Heightman, James F Callahan, Elisabetta Chiarparin

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Frequent Collaborators

3 joint publications

Paul N Mortenson

3 joint publications

Alison J-A Woolford

3 joint publications

Jeffrey K Kerns

2 joint publications

Tom D Heightman