Hironori Hayashi
9PUBLICATIONS
42CO-AUTHORS

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Publications (9)
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|Jan 20, 2025
An orally available P1'-5-fluorinated Mpro inhibitor blocks SARS-CoV-2 replication without booster and exhibits high genetic barrier.Nobuyo Higashi-Kuwata, Haydar Bulut, Hironori Hayashi
|Sep 05, 2024
Structural and virologic mechanism of the emergence of resistance to Mpro inhibitors in SARS-CoV-2.Shin-Ichiro Hattori, Haydar Bulut, Hironori Hayashi
|Feb 09, 2024
Helix-based screening with structure prediction using artificial intelligence has potential for the rapid development of peptide inhibitors targeting class I viral fusion.Satoshi Suzuki, Mio Kuroda, Keisuke Aoki
|Jul 12, 2023
GRL-142 binds to and impairs HIV-1 integrase nuclear localization signal and potently suppresses highly INSTI-resistant HIV-1 variants.Manabu Aoki, Hiromi Aoki-Ogata, Haydar Bulut
|Feb 25, 2023
Identification of SARS-CoV-2 Mpro inhibitors containing P1' 4-fluorobenzothiazole moiety highly active against SARS-CoV-2.Nobuyo Higashi-Kuwata, Kohei Tsuji, Hironori Hayashi
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Frequent Collaborators
4 joint publications
Haydar Bulut
4 joint publications
Kazuya Hasegawa
4 joint publications
Nobutoki Takamune
4 joint publications
Shin-Ichiro Hattori
3 joint publications
Manabu Aoki
3 joint publications
Debananda Das
3 joint publications
Nobuyo Higashi-Kuwata
3 joint publications
Shogo Misumi
3 joint publications
Hiromi Ogata-Aoki
3 joint publications
Naoki Kishimoto