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Christopher Wellaway

9PUBLICATIONS

64CO-AUTHORS

Genome structure and regulationBiologically active moleculesBiomaterialsHaematological tumoursNonlinear optics and spectroscopy

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Publications (9)

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|Jun 12, 2024

Structure- and Property-Based Optimization of Efficient Pan-Bromodomain and Extra Terminal Inhibitors to Identify Oral and Intravenous Candidate I-BET787.

David J Hirst, Paul Bamborough, Niam Al-Mahdi

|Nov 15, 2023

Structure-Guided Design of a Domain-Selective Bromodomain and Extra Terminal N-Terminal Bromodomain Chemical Probe.

Erin Bradley, Lucia Fusani, Chun-Wa Chung

|Jan 07, 2022

Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate.

Philip G Humphreys, Stephen J Atkinson, Paul Bamborough

|Dec 20, 2021

Investigation of Janus Kinase (JAK) Inhibitors for Lung Delivery and the Importance of Aldehyde Oxidase Metabolism.

Christopher R Wellaway, Ian R Baldwin, Paul Bamborough

|Aug 14, 2020

Structure-Based Design of a Bromodomain and Extraterminal Domain (BET) Inhibitor Selective for the N-Terminal Bromodomains That Retains an Anti-inflammatory and Antiproliferative Phenotype.

Christopher R Wellaway, Paul Bamborough, Sharon G Bernard

|Mar 21, 2020

Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation.

Omer Gilan, Inmaculada Rioja, Kathy Knezevic

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Frequent Collaborators

6 joint publications

Paul Bamborough

6 joint publications

Chun-Wa Chung

4 joint publications

Philip G Humphreys

3 joint publications

Rishi R Shah

2 joint publications

Johanna Vappiani

2 joint publications

Enid Y N Lam

2 joint publications

Paola Grandi

2 joint publications

Thilo Werner

2 joint publications

Mark A Dawson

2 joint publications

Rab K Prinjha

Frequent Collaborators

6 joint publications

Paul Bamborough

6 joint publications

Chun-Wa Chung

4 joint publications

Philip G Humphreys

3 joint publications

Rishi R Shah

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