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Rishi R Shah

6PUBLICATIONS
22CO-AUTHORS
Pharmaceutical delivery technologiesMedical devicesBiologically active molecules
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Journal

Publications (6)

Sort by Publication Date:
|Mar 08, 2025
Challenges, opportunities, and therapeutic potential of JAK inhibitors and their derived PROTACs (2022 - 2023).

Rishi R Shah

|Mar 13, 2024
Structure-Guided Design and Optimization of Covalent VHL-Targeted Sulfonyl Fluoride PROTACs.

Rishi R Shah, Elena De Vita, Preethi S Sathyamurthi

|Nov 15, 2023
Structure-Guided Design of a Domain-Selective Bromodomain and Extra Terminal N-Terminal Bromodomain Chemical Probe.

Erin Bradley, Lucia Fusani, Chun-Wa Chung

|Nov 15, 2022
Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432.

Philip G Humphreys, Niall A Anderson, Paul Bamborough

|Dec 20, 2021
Investigation of Janus Kinase (JAK) Inhibitors for Lung Delivery and the Importance of Aldehyde Oxidase Metabolism.

Christopher R Wellaway, Ian R Baldwin, Paul Bamborough

|Jan 07, 2020
Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening.

Christopher R Wellaway, Dominique Amans, Paul Bamborough

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Frequent Collaborators

3 joint publications

Christopher R Wellaway

3 joint publications

Paul Bamborough

3 joint publications

Philip G Humphreys

3 joint publications

Chun-Wa Chung

1 joint publications

David J Hirst

1 joint publications

Francesco Rianjongdee

1 joint publications

Niall A Anderson

1 joint publications

Toryn Dalton

1 joint publications

Julie C L Fournier

1 joint publications

Heather F Gray

Frequent Collaborators

3 joint publications

Christopher R Wellaway

3 joint publications

Paul Bamborough

3 joint publications

Philip G Humphreys

3 joint publications

Chun-Wa Chung

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