Katherine L Jones

5PUBLICATIONS
18CO-AUTHORS
Cheminformatics and quantitative structure-activity relationshipsMolecular targetsGenome structure and regulationMedical devices
Featured researcher

Get your video featured.

JoVEPublish with JoVE
Journal

Publications (5)

|Aug 20, 2026
Structure-Activity Relationship Studies Resulting in the Identification of Potent and Selective Salt-Inducible Kinase Inhibitors.

|May 04, 2026
Targeting Activin Receptor-like Kinase 2 Using Heterobifunctional Protein Degraders.

|Jun 12, 2024
Structure- and Property-Based Optimization of Efficient Pan-Bromodomain and Extra Terminal Inhibitors to Identify Oral and Intravenous Candidate I-BET787.

David J Hirst, Paul Bamborough, Niam Al-Mahdi

|Nov 15, 2022
Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432.

Philip G Humphreys, Niall A Anderson, Paul Bamborough

|Aug 13, 2021
Discovery of a Novel Bromodomain and Extra Terminal Domain (BET) Protein Inhibitor, I-BET282E, Suitable for Clinical Progression.

Katherine L Jones, Dominic M Beaumont, Sharon G Bernard

Pageof 1

Frequent Collaborators

3 joint publications

Chun-Wa Chung

2 joint publications

Philip G Humphreys

2 joint publications

Paul Bamborough

2 joint publications

William J Kerr