Shaun M Fillery
7PUBLICATIONS
19CO-AUTHORS
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Publications (7)
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|Jul 03, 2023
Discovery of AZD4747, a Potent and Selective Inhibitor of Mutant GTPase KRASG12C with Demonstrable CNS Penetration.Jason G Kettle, Sharan K Bagal, Derek Barratt
|Apr 26, 2022
Discovery of AZD4625, a Covalent Allosteric Inhibitor of the Mutant GTPase KRASG12C.Jason G Kettle, Sharan K Bagal, Sue Bickerton
|Feb 08, 2022
Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models.Jon J Winter-Holt, Catherine Bardelle, Elisabetta Chiarparin
|Nov 22, 2021
Diverse, Potent, and Efficacious Inhibitors That Target the EED Subunit of the Polycomb Repressive Complex 2 Methyltransferase.Sharan K Bagal, Clare Gregson, Daniel H O' Donovan
|Jul 25, 2020
A Buchwald-Hartwig Protocol to Enable Rapid Linker Exploration of Cereblon E3-Ligase PROTACs*.Thomas G Hayhow, Rachel E A Borrows, Coura R Diène
|Feb 06, 2020
Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRASG12C.Jason G Kettle, Sharan K Bagal, Sue Bickerton
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Frequent Collaborators
3 joint publications
Jason G Kettle
3 joint publications
Michael S Bodnarchuk
3 joint publications
Frederick W Goldberg
3 joint publications
Graeme Robb
2 joint publications
Doyle J Cassar
2 joint publications
Hilary J Lewis
1 joint publications
Rodrigo J Carbajo
1 joint publications
Miguel A Cortés González
1 joint publications
Magnus Schou
1 joint publications
Thomas G Hayhow
